l-Menthol (CAS 2216-51-5) — Citrus Top-Middle Note Fragrance Ingredient

Citrus · Spicy

l-Menthol

CAS 2216-51-5

Origin
synthetic
Note
Top-Middle
IFRA
Generally safe
Data as of: Apr 2026

What Is l-Menthol?

l-Menthol is the naturally occurring form of menthol, most commonly associated with the cooling sensation in peppermint and mint products. You’ll encounter it in chewing gum, toothpaste, cough drops, and topical pain relievers. This enantiomer provides superior cooling effects compared to synthetic racemic mixtures, making it prized in both flavor and fragrance applications.

Safety Profile

GENERALLY SAFE
Generally safeUse with awarenessProfessional use
GRAS status for food use
Avoid high concentrations on sensitive skin
CAS
2216-51-5
Formula
Mixture
MW
Variable
Odor Family
Citrus · Spicy
Layer 1 · Enthusiast

What Does l-Menthol Smell Like?

l-Menthol bursts with an intense, crystalline freshness – like Arctic wind blowing through a peppermint field. The initial sensation is sharply cooling, almost painful in its purity, before mellowing into a rounded herbal sweetness. Unlike synthetic menthols, it maintains a clean, natural character throughout evaporation without chemical harshness. The dry-down reveals subtle woody undertones that prevent the cooling effect from becoming clinical or medicinal.

Scent Profile

In Famous Fragrances

Fragrance associations may not reflect actual formulations.

Cool Water(Davidoff, 1988)

Used sparingly to amplify the aquatic freshness with its natural cooling properties, creating the illusion of ocean breezes without overt mintiness.

Green Irish Tweed(Creed, 1985)

Provides subtle cooling contrast to the violet leaf and iris, enhancing the dew-on-grass freshness of this classic fougère.

Layer 2

2D Molecular Structure

(1R,2S,5R)-(-)-Menthol

SMILES: CC(C)[C@@H]1CC[C@@H](C)C[C@H]1O

Chemistry, Properties & Perfumer Guide

The Chemistry

l-Menthol is a monoterpenoid alcohol with three chiral centers, occurring naturally in Mentha arvensis and other mint species. The (-)-menthol enantiomer binds preferentially to TRPM8 cold receptors, explaining its superior cooling effect. Industrial production typically involves hydrogenation of thymol or resolution of racemic menthol mixtures. The L-form crystallizes in characteristic hexagonal plates due to its specific molecular geometry.

Physical & Chemical Properties

Melting Point42-45 °C
Boiling Point212 °C
Optical Rotation-50° (c=10, ethanol)

Perfumer Guide

Note Position
Top-Middle
Volatility
Moderate (2-4 hours)
Blending
Good with citrus, challenging with florals
ApplicationTypical %RangeNotes
Fine Fragrance0.1-0.5%Up to 1%Cooling accent
Functional Fragrance0.5-2%Up to 5%Freshness booster

Classic Accords

+ Eucalyptus + Camphor = Medicinal + Lime + Basil = Mojito + Vanilla + Tonka = Ice Cream

Tip: Balance cooling effects with warm base notes to prevent fragrance from feeling clinical.

Alternatives & Comparisons

1
Racemic Menthol CAS 89-78-1

Less expensive but weaker cooling effect; use when cost is prioritized over performance.

2
WS-3 CAS 39711-79-0

Synthetic coolant without mint odor for applications requiring pure cooling sensation.

Layer 3

Safety, Regulatory & Sustainability

⚠ Regulatory Disclaimer

General reference only. Consult current IFRA Standards Library before formulating.

IFRA Status

No IFRA restrictions. Approved for all fragrance categories.

RIFM Assessment

Considered safe for current use levels in fragrance applications.

Sustainability

Most l-menthol is now produced synthetically from renewable turpentine feedstocks, reducing pressure on wild mint populations. The L-enantiomer’s higher potency means less material is required compared to racemic mixtures, improving sustainability metrics.

Explore l-Menthol

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References

  1. Eccles R. (1994). Menthol and related cooling compounds. Journal of Pharmacy and Pharmacology. PMID 7932039

Data: PubChem (NIH), PubMed, RIFM, IFRA. Last reviewed: Apr 2026.

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Physicochemical Properties

DTXSID: DTXSID1022180

Physical Properties

Molecular Weight 156.269 g/mol🔬 EPA CompTox
Density 0.49 g/cm^3🔬 EPA CTX
Boiling Point 214.254 °C📊 OPERA
Melting Point 42.931 °C🔬 EPA CTX
Flash Point 92.825 °C🔬 EPA CTX
Refractive Index 1.457 Dimensionless📊 OPERA
Molar Volume 175.542 cm^3/mol📊 OPERA

Partition & Solubility

LogP (Octanol-Water) 3.256 Log10 unitless🔬 EPA CTX
LogD (pH 5.5) 3.242 Log10 unitless📊 OPERA
LogD (pH 7.4) 3.242 Log10 unitless📊 OPERA
LogKoa (Octanol-Air) 6.6 Log10 unitless📊 OPERA
Water Solubility 0.003 mol/L🔬 EPA CTX
Henry's Law Constant 0 atm-m3/mole📊 OPERA

Transport Properties

Vapor Pressure 0.12 mmHg🔬 EPA CTX
Viscosity 9.449 cP📊 OPERA
Surface Tension 29.625 dyn/cm📊 OPERA
Thermal Conductivity 129.72 mW/(m*K)📊 OPERA

Molecular Descriptors

Topological Polar Surface Area 20.23 Ų💻 Computed
H-Bond Donors 1 count💻 Computed
H-Bond Acceptors 1 count💻 Computed
Rotatable Bonds 1 count💻 Computed
Aromatic Rings 0 count💻 Computed
Molar Refractivity 47.833 cm^3/mol📊 OPERA
Polarizability 18.963 Å^3📊 OPERA

Data Sources:

🔬 EPA Experimental data from U.S. EPA CompTox Chemicals Dashboard & CTX APIs. 📊 OPERA Predicted using EPA's OPERA QSAR models. 💻 Computed Calculated from SMILES using RDKit.

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